Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Adenosine A1 receptor activator T62 是腺苷 A1 受体的变构增强剂,有镇痛作用。
规格 | 价格/CNY | 货期 | 数量 | |
---|---|---|---|---|
1 mg | ¥ 1,190 | 现货 | ||
5 mg | ¥ 3,230 | 现货 | ||
10 mg | ¥ 4,630 | 现货 | ||
25 mg | ¥ 7,150 | 现货 | ||
50 mg | ¥ 9,630 | 现货 | ||
100 mg | ¥ 12,800 | 现货 | ||
500 mg | ¥ 25,800 | 现货 | ||
1 mL * 10 mM (in DMSO) | ¥ 2,730 | 现货 |
产品描述 | Adenosine A1 receptor activator T62 is an allosteric enhancer of adenosine A1 receptor, and it produces antinociception in animal models of acute pain and also reduces hypersensitivity in models of inflammatory and nerve-injury pain[1][2][3]. |
体内活性 | Adenosine A1 receptor activator T62 (0.3-3 μg; intrathecal administration; male SpragueDawley rats) treatment produces a dose-dependent antihypersensitivity effect. However it has no effect on ambulation or activity level[1]. |
动物实验 | Intrathecal T62 of Male SpragueDawley rats (250 g) after paw incision surgery with the dose of 0.3 μg, 0.5 μg, 1 μg, and 3 μg, produced a dose-dependent antihypersensitivity effect, with no effect on ambulation or activity level. The ED40 (95% confidence interval) for T62 was 0.77 (0.63-0.91) microg. |
分子量 | 291.8 |
分子式 | C15H14ClNOS |
CAS No. | 40312-34-3 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 75 mg/ml (257.03 mM)
可选溶剂 | 浓度 体积 质量 | 1 mg | 5 mg | 10 mg | 25 mg |
DMSO | 1 mM | 3.427 mL | 17.135 mL | 34.27 mL | 85.6751 mL |
5 mM | 0.6854 mL | 3.427 mL | 6.854 mL | 17.135 mL | |
10 mM | 0.3427 mL | 1.7135 mL | 3.427 mL | 8.5675 mL | |
20 mM | 0.1714 mL | 0.8568 mL | 1.7135 mL | 4.2838 mL | |
50 mM | 0.0685 mL | 0.3427 mL | 0.6854 mL | 1.7135 mL | |
100 mM | 0.0343 mL | 0.1714 mL | 0.3427 mL | 0.8568 mL |
对于不同动物的给药剂量换算,您也可以参考 更多...
请在以下方框中输入您的动物实验信息后点击计算,可以得到母液配置方法和体内配方的制备方法: 比如您的给药剂量是10 mg/kg,每只动物体重20 g,给药体积100 μL,一共给药动物10 只,您使用的配方为5% DMSO+30% PEG300+5% Tween 80+60% ddH2O。那么您的工作液浓度为2 mg/mL。
母液配置方法:2 mg 药物溶于 50 μL DMSO (母液浓度为 40 mg/mL), 如您需要配置的浓度超过该产品的溶解度,请先与我们联系。
体内配方的制备方法:取 50 μL DMSO 主液,加入 300 μL PEG300, 混匀澄清,再加 50 μL Tween 80,混匀澄清,再加 600 μL ddH2O, 混匀澄清。
您可能有的问题的答案可以在抑制剂处理说明中找到,包括如何准备库存溶液,如何存储产品,以及基于细胞的分析和动物实验需要特别注意的问题。
Adenosine A1 receptor activator T62 40312-34-3 GPCR/G Protein Neuroscience Adenosine Receptor allosteric Inhibitor P1 receptor adenosine hypersensitivity α2-adrenoceptors antihypersensitivity intrathecal Enhancer neuropathic Adenosine A-1 receptor activator T62 inhibit inhibitor